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Dec, 2023
DTIAM: 一个统一的框架用于预测药物靶标相互作用、结合亲和力和激活/抑制机制
DTIAM: A unified framework for predicting drug-target interactions, binding affinities and activation/inhibition mechanisms
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Zhangli Lu, Chuqi Lei, Kaili Wang, Libo Qin, Jing Tang...
TL;DR
DTIAM提供了一个统一的框架,可准确而可靠地预测药物靶点相互作用、结合亲和性和激活/抑制机制。
Abstract
Accurate and robust
prediction
of
drug-target interactions
(DTIs) plays a vital role in drug discovery. Despite extensive efforts have been invested in predicting novel DTIs, existing approaches still suffer from
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